Decarboxylative Coupling Reaction of 2‐(1 H ‐Indol‐3‐yl)acetic Acids with Indole, Azaindole, Benzimidazole and Indazole Derivatives
نویسندگان
چکیده
منابع مشابه
Suzuki-Miyaura cross-coupling of unprotected, nitrogen-rich heterocycles: substrate scope and mechanistic investigation.
The Suzuki-Miyaura cross-coupling of unprotected, nitrogen-rich heterocycles using precatalysts P1 or P2 is reported. The procedure allows for the reaction of variously substituted indazole, benzimidazole, pyrazole, indole, oxindole, and azaindole halides under mild conditions in good to excellent yields. Additionally, the mechanism behind the inhibitory effect of unprotected azoles on Pd-catal...
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ژورنال
عنوان ژورنال: Advanced Synthesis & Catalysis
سال: 2019
ISSN: 1615-4150,1615-4169
DOI: 10.1002/adsc.201900688